APIs intermediates |
|
PRODUCT NAME |
CAS No. |
1 |
Quetiapine |
2-(2-chloroethoxy)ethanol |
628-89-7 |
2 |
2-(2-hydroxyethoxy)ethyl)piperazine |
13349-82-1 |
3 |
dibenzo[b,f][1,4]thiazepine-11-[10H]one |
3159-07-7 |
4 |
Gefitinib |
4-(3-chloro-4-fluorophenylamino)-7-methoxyquinazolin-6-ol |
184475-71-6 |
5 |
6-hydroxy-7-methoxy-3,4-dihydroquinazolin-4(3H)-one |
179688-52-9 |
6 |
6-acetoxy-7-methoxy-3,4-dihydroquinazolin-4(3H)-one |
179688-53-0 |
7 |
7-methoxy-6-(3-morpholin-4-ylpropoxy)quinazolin-4(3H)-one |
199327-61-2 |
8 |
Erlotinib |
3,4-bis(2-methoxyethoxy)benzoic acid ethyl ester |
183322-16-9 |
9 |
ethyl 2-amino-4,5-bis(2-methoxyethoxy)-2-aminobenzoate |
950596-58-4 |
10 |
6,7-bis-(2-methoxyethoxy)-quinazolin-4(3H)-one |
179688-29-0 |
11 |
4-chloro-6,7-di(2-methoxyethoxy)quinazoline |
183322-18-1 |
12 |
Lapatinib |
3-chloro-4-(3-fluorobenzyloxy)nitrobenzene |
443882-99-3 |
13 |
3-chloro-4-(3-fluorobenzyloxy)aniline |
202197-26-0 |
14 |
4-chloro-6-iodoquinazoline |
98556-31-1 |
15 |
2-aminoethylmethylsulfone hydrochloride |
104458-24-4 |
16 |
2-formylfuran-5-boronic acid |
27329-70-0 |
17 |
6-iodoquinazolin-4-one |
16064-08-7 |
18 |
N-[3-chloro-4-(3-fluorobenzyloxy)phenyl]-6-iodoquinazolin-4-amine |
231278-20-9 |
19 |
Sorafenib |
4-chloro-pyridine-2-carbonyl chloride |
53750-66-6 |
20 |
4-(4-aminophenoxy)-N-methylpicolinamide |
284462-37-9 |
21 |
N-methyl-4-chloropyridine-2-carboxamide |
220000-87-3 |
22 |
Imatinib |
4-[(4-methylpiperazin-1-yl)methyl]benzoic acid dihydrochloride |
106261-49-8 |
23 |
N-(5-amino-2-methylphenyl)-4-(3-pyridyl)-2-pyrimidineamine |
152460-10-1 |
24 |
Raloxifene |
N-(2-(4-bromophenoxy)ethyl)piperidine hydrochloride |
399016-75-2 |
25 |
Sunitinib |
5-formyl-2,4-dimethyl-1H-pyrrole-3-carboxylic acid |
253870-02-9 |
26 |
ethyl 2,4-dimethyl-1H-pyrrole-3-carboxylate |
2199-51-1 |
27 |
4-(ethoxycarbonyl)-3,5-dimethyl-1H-pyrrole-2-carboxylic acid |
5442-91-1 |
28 |
ethyl 5-formyl-2,4-dimethyl-1H-pyrrole-3-carboxylate |
2199-59-9 |
29 |
N-(2-(diethylamino)ethyl)-5-formyl-2,4-dimethyl-1H-pyrrole-3-carboxamide |
356068-86-5 |
30 |
Dasatinib |
2-amino-N-(2-chloro-6-methylphenyl)thiazole-5-carboxamide |
302964-24-5 |
31 |
(E)-N-(2-chloro-6-methylphenyl)-3-ethoxyacrylamide |
863127-76-8 |
32 |
2-(6-chloro-2-methylpyrimidin-4-ylamino)-N-(2-chloro-6- methylphenyl) thiazole-5-carboxamide |
302964-08-5 |
33 |
Nilotinib |
4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]benzoic acid |
641569-94-0 |
34 |
4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]benzoic acid ethyl ester |
641569-97-3 |
35 |
3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)aniline |
641571-11-1 |
36 |
Bosutinib |
1-(3-chloropropyl)-4-methylpiperazine dihydrochloride |
2031-23-4 |
37 |
3-(3-(4-methylpiperazinyl)propoxy)-4-methoxyaniline |
|
38 |
Pazopanib |
3-methyl-6-nitroindazole |
6494-19-5 |
39 |
2,3-dimethyl-2H-indazol-6-amine HCl |
635702-60-2 |
40 |
3-amino-6-methylbenzenesulfonamide |
6973-9-7 |
41 |
Dronedarone |
N-(3-chloropropyl)dibutylamine |
36421-15-5 |
42 |
Ticagrelor |
2-chloro-1-(3,4-difluoro-phenyl)-ethanone |
51336-95-9 |
43 |
Fluvastatin |
N-isopropylaniline |
768-52-5 |
44 |
3-(4-fluorophenyl)-1-isopropyl-1H-indole |
93957-49-4 |
45 |
3-(N-phenyl-N-methyl)aminoacrolein |
14189-82-3 |
46 |
3-[3-(4-fluorophenyl)-1-(1-methylethyl)-1H-indol-2-yl]-(E)-2-propenal |
93957-50-7 |
47 |
Ritonavir |
carbonic acid 4-nitrophenyl 5-thiazolylmethyl ester |
144163-97-3 |
48 |
1-(2-isopropylthiazol-4-yl)-N-methylmethanamine dihydrochloride |
908591-25-3 |
49 |
N-[N-methyl-N-((2-isopropyl-4-thiazolyl)methyl)aminocarbonyl]-L-valine lithium salt |
201409-23-6 |
50 |
N-((N-methyl-N-((2-isopropyl-4-thiazolyl)methyl)amino)carbonyl)-L-valine |
154212-61-0 |
51 |
Pentoxyverine |
2-(2-(diethylamino)ethoxy)ethanol |
140-82-9 |
52 |
Fluvoxamine |
(4-trifluoromethyl)-5-methoxyvalerophenone |
61718-80-7 |
53 |
Apixaban |
ethyl 2-chloro-2-(2-(4-methoxyphenyl) hydrazono)acetate |
27143-07-3 |
54 |
3-chloro-1-(4-nitrophenyl)-5,6-dihydropyridin-2(1H)-one |
536760-29-9 |
55 |
3-morpholino-1-(4-(2-oxopiperidin-1-yl)phenyl)-5,6-dihydropyridin-2(1H)-one |
545445-44-1 |
56 |
Lamivudine |
(1R,2S,5R)-menthyl-(2R,5S)-5-(4-amino-2-oxo-2H-pyrimidin-1-yl)-[1,3]oxathiolane-2-carboxylic acid |
147027-10-9 |
57 |
Dirithromycin |
1,1-dimethoxy-2-(2-methoxyethoxy)ethane |
94158-44-8 |
58 |
Trazodone |
1-(3-chlorophenyl)-4-(3-chloropropyl)piperazine hydrochloride |
39577-43-0 |
59 |
Carvedilol |
2-(2-methoxyphenoxy)ethylamine |
1836-62-0 |
60 |
Tamsulosin |
2-(2-ethoxyphenoxy)ethylamine |
6781-17-5 |
61 |
Iloperidone |
4-(3-chloropropoxy)-3-methoxyacetophenone |
58113-30-7 |
62 |
Parecoxib Sodium |
3,4-diphenyl-5-methylisoxazole |
37928-17-9 |
63 |
Terbinafine |
1-chloro-6,6-dimethyl-2-hepten-4-yne |
126764-17-8 |
64 |
1-methyl-aminomethyl naphthalene |
14489-75-9 |
65 |
N-methyl-1-naphthalenemethylamine hydrochloride |
65473-13-4 |
66 |
Linezolid |
3-fluoro-4-morpholin--4-yl-phenylamine |
93246-53-8 |
67 |
N-benzyloxycarbonyl-3-fluoro-4-morpholinoaniline |
168828-81-7 |
68 |
Dabigatran etexilate |
ethyl 3-(pyridin-2-ylamino)propanoate |
103041-38-9 |
69 |
ethyl 3-(3-amino-4-(methylamino)-N-(pyridin-2-yl)benzamido)propanoate |
212322-56-0 |
70 |
Rosiglitazon |
2-N-methyl-2-pyridylaminoethanol |
122321-04-4 |
71 |
Emtricitabine |
5-fluorocystosine |
2022-85-7 |
72 |
Vilazodone |
ethyl 5-(piperazin-1-yl) benzofuran-2-carboxylate |
163521-20-8 |
73 |
5-(piperazin-1-yl)benzofuran-2-carboxamide |
183288-46-2 |
74 |
tert-butyl 4-(2-carbamoylbenzofuran-5-yl)piperazine-1-carboxylate |
183288-44-0 |